Bromobenzenes
Selleck Chemical LLC AZ3451-5mg
AZ3451 is a potent antagonist of protease-activated receptor 2 (PAR2) that binds to a remote allosteric site outside the helical bundle with IC50 of 23 nM.
Selleck Chemical LLC IDO-IN-2
IDO-IN-2 (RG 6078 NLG-919 analogue GDC-0919 analogue) is a a potent IDO1 inhibitor with IC50 of 38 nM
Selleck Chemical LLC 1-Azakenpaullone
1-Azakenpaullone (1-Akp) is a potent and selective GSK-3 inhibitor with IC50 of 18 nM 100-fold selectivity over CDK1/cyclin B and CDK5/p25
Selleck Chemical LLC CCT020312-E1030-5MG
CCT020312 is a selective PERK (EIF2AK3) activator with an EC50 of 5 1 M CCT020312 can be used for the selective activation of EIF2A-mediated translation control
Selleck Chemical LLC Histone Acetyltransferase Inhibitor II S1161-5mg
Histone Acetyltransferase Inhibitor II (HAT Inhibitor II compound 2c) is a potent selective and cell-permeable p300 histone acetyltransferase (HAT) inhibitor with IC50 of 5 M Histone Acetyltransferase Inhibitor II shows anti-acetylase activity in mammalian cells
Selleck Chemical LLC P7C3-10mg
P7C3 is a potent proneurogenic and neuroprotective chemical that targets NAMPT enzyme.
Selleck Chemical LLC BIO-acetoxime-5mg
BIO-acetoxime (GSK-3 Inhibitor X) is a potent dual GSK3α/β inhibitor with IC50 of 10 nM, >240-fold selectivity over CDK5/p25, CDK2/cyclin A and CDK1/cyclin B.
Selleck Chemical LLC H 89 2HCl S1582-200mg
H 89 2HCl is a potent PKA inhibitor with Ki of 48 nM in a cell-free assay 10-fold selective for PKA than PKG 500-fold greater selectivity than PKC MLCK calmodulin kinase II and casein kinase I/II H 89 2HCl induces autophagy
Selleck Chemical LLC IDO-IN-1
IDO-IN-1 is a potent indoleamine 2 3-dioxygenase (IDO) inhibitor with an IC50 of 59 nM
Selleck Chemical LLC Kenpaullone-5mg
Kenpaullone (9-Bromopaullone, NSC-664704) is an ATP-competitive inhibitor of cyclin-dependent kinases (CDKs). It also inhibit glycogen synthase kinase 3β (GSK3β) with IC50 of 0.23 µM.
Selleck Chemical LLC BCI-121-5mg
BCI-121 is a potent inhibitor of SMYD3 that impairs the proliferation of many kinds of cancer cells.
Medchemexpress LLC eIF4A3-IN-8 | 18474-59-4 | 99.9% | 175.18 | 100 MG
eIF4A3-IN-8 is a selective ATP-competitive eukaryotic initiation factor 4A3 (eIF4A3) inhibitor. It can serve as a valuable chemical probe to elucidate the detailed function of eIF4A3 and the exon junction complex (EJC).
- Selective ATP-competitive inhibitor
- Chemical probe for elucidating eIF4A3 and EJC function
![Medchemexpress LLC 4H-1-benzothiopyran-4-one, 2,3-dihydro-2-[1-(phenylmethyl)-4-piperidinyl]- | 1204401-49-9 | MFCD18206882 | 99.9% | 337.48 g/mol | C21H23NOS | 10 MG](https://assets.fishersci.com/TFS-Assets/CCG/product-images/5000242751.png-250.jpg)
Medchemexpress LLC 4H-1-benzothiopyran-4-one, 2,3-dihydro-2-[1-(phenylmethyl)-4-piperidinyl]- | 1204401-49-9 | MFCD18206882 | 99.9% | 337.48 g/mol | C21H23NOS | 10 MG
σ1 Receptor antagonist-1 is a potent and selective sigma-1 receptor antagonist provided as a solid research chemical for in vitro studies. It has high reported affinity for the σ1 receptor and has been used in cell-based assays to inhibit cell growth, induce apoptosis, and arrest the cell cycle. Analytical data and handling information are provided by the supplier; this compound is for research use only.
Medchemexpress LLC σ1 receptor antagonist-1 | 1204401-49-9 | MFCD18206882 | 99.9% | 337.48 g/mol | C21H23NOS | 50 MG
σ1 Receptor antagonist-1 is a small-molecule sigma-1 receptor antagonist supplied for laboratory research use. It is provided as a light yellow to light brown solid with high chemical purity, characterized by molecular formula C21H23NOS and molecular weight 337.48 g/mol. Recommended storage conditions differ for powder and solution forms; handle per safety data sheet.
Medchemexpress LLC BCI hydrochloride 5mg | 95130-23-7 | 5 MG
BCI hydrochloride is the hydrochloride salt of (E)-BCI, a small-molecule inhibitor of dual-specificity phosphatases DUSP6 and DUSP1. It is supplied as a solid research reagent for biochemical and cell-based studies to modulate MAPK pathway signalling.
- Selective DUSP6 and DUSP1 inhibitor useful for MAPK pathway studies.
- High chemical purity (99.93% as listed by the supplier).
- Solid form, suitable for storage and dissolution in common solvents.
- Supplied in a 5 MG quantity for small-scale laboratory research.
- Identified by CAS 95130-23-7 for unambiguous compound reference.